Gravett, Edward C., Hilton, Philip J, Jones, Keith and Peron, Jean-Marie (2003) A new route to 5-aryl and 5-heteroaryl-2-pyrones via Suzuki coupling of a 2-pyrone-5-boronate ester. Synlett, 2, 0253-0255. ISSN (print) 0936-5214Full text not available from this archive.
A synthesis of boronate (III) is reported along with its use in Pd-catalyzed coupling reactions with aryl halides and triflates. Catalytic hydrogenation of the resulting products provides a rapid way of introducing a valerolactone residue onto an aromatic ring.
|Uncontrolled Keywords:||Suzuki coupling, palladium, boron, heterocycles, pyrone, radicals|
|Faculty, School or Research Centre:||Faculty of Science (until 2011) > School of Pharmacy and Chemistry|
|Depositing User:||Jean-Marie Peron|
|Date Deposited:||12 Nov 2010 10:59|
|Last Modified:||12 Jan 2011 14:13|
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